Triptorelin IUPAC nomenclature 5-oxo-D-prolyl-L-histidyl-Ltryptophyl-L-seryl-Ltyrosyl-3-(1H-indol-2-yl)-L-alanylleucyl-L-arginyl-L-prolylglycinamide. Classification Triptorelin is a GnRH analogue. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 1311.4 g/mol 2 Physical appearance White to off white powder. Present in salt form as triptorelin pamoate […]
Finasteride IUPAC nomenclature (1S,3aS,3bS,5aR,9aR,9bS,11aS)-N-tert-butyl-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,5a,6,9b,10,11-dodecahydroindeno[5,4-f]quinoline-1-carboxamide. Classification Finasteride is a 5-α reductase inhibitor. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 372.5g/mol 2 Appearance Fine white to off white crystalline solid 3 Melting point 252-254°C 4 Solubility […]
Dutasteride IUPAC nomenclature (1S,3aS,3bS,5aR,9aR,9bS,11aS)-N-[2,5-bis(trifluoromethyl)phenyl]-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,5a,6,9b,10,11-dodecahydroindeno[5,4-f]quinoline-1-carboxamide. Classification Dutasteride is a 5-α reductase inhibitor. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 528.5 g/mol 2 Appearance Solid 3 Melting point 242-250°C 4 Solubility Insoluble 5 Octanol/water partition coefficient 6.8 […]
Nafarelin IUPAC nomenclature (2R)-N-[(2R)-5-carbamimidamido-1-[(2S)-2-[(carbamoylmethyl)carbamoyl]pyrrolidin-1-yl]-1-oxopentan-2-yl]-2-[(2R)-2-[(2R)-2-[(2R)-3-hydroxy-2-[(2S)-2-[(2S)-3-(1H-imidazol-4-yl)-2-{[(2R)-5-oxopyrrolidin-2-yl]formamido}propanamido]-3-(1H-indol-3-yl)propanamido]propanamido]-3-(4-hydroxyphenyl)propanamido]-3-(naphthalen-2-yl)propanamido]-4-methylpentanamide. Classification Nafarelin is a GnRH analogue. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 1322.5 g/mol 2 Appearance White to off white solid 3 Melting point More than 181°C 4 Solubility […]
Bicalutamide IUPAC nomenclature (RS)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorophenyl)sulfonyl]-2-hydroxy-2-methylpropanamide. Classification Bicalutamide is an antiandrogen. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 430.4 g/mol 2 Appearance Fine white to off white powder 3 Melting point 191-193°C 4 Solubility Soluble in […]
Letrozole IUPAC nomenclature 4,4′-((1H-1,2,4-triazol-1-yl)methylene)dibenzonitrile. Classification Letrozole is an aromatase inhibitor. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 285.3 g/mol 2 Appearance White to yellow crystalline powder. It is present in anhydrous crystal form 3 […]
Fulvestrant IUPAC nomenclature (7R,8R,9S,13S,14S,17S)-13-methyl-7-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-3,17-diol. Classification Fulvestrant is a selective estrogen receptor down regulator. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 606.8 g/mol 2 Appearance Present as white powder form. The solution for injection appears […]
Toremifene IUPAC nomenclature 2-[4-[(1Z)-4-Chloro-1,2-diphenyl-but-1-en-1-yl]phenoxy]-N,N-dimethylethanamine. Classification Toremifene is a selective estrogen receptor modulator. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 406 g/mol 2 Appearance Present in the solid form 3 Melting point 108-110°C 4 […]
Ethinylestradiol IUPAC nomenclature (8R,9S,13S,14S,17R)-17-ethynyl-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diol. Classification Ethinylestradiol is classified as an estrogen drug, altering the hormonal milieu. [1] Physiochemical Properties S. NO. PHYSICAL AND CHEMICAL PROPERTIES 1 Molecular weight 296.4 g/mol 2 Appearance White to creamy white powder 3 Melting point […]